Full 2L QBank
Pharmacology General pharmacology c714750a

Paial agonist can antagonise the effects of a full agonist because it has

A
High affinity but low intrinsic activity
B
No affinity and low intrinsic activity
C
Low affinity but high intrinsic activity
D
High affinity but no intrinsic activity
High-Yield Explanation
Agonists:- Have both affinity and maximal intrin-sic activity. Competitive antagonists :- Have affinity but no intrinsic activity. Paial agonists:- Have affinity and submaximal intrinsic activity. Inverse agonists:- Have affinity but intrinsic activity with a minus sign (IA between 0 and -1). Ref:- kd tripathi; pg num:-41,42

Related Pharmacology MCQs

Practice 2,00,000+ NEET PG Questions Free

Timed mock tests, mistake queue analytics, audio lectures & zero attempt limits on i❤️Exams.

Start Free Mock Test Now