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Pharmacology General 9ce77597

Inverse agonist is -

A
Buspirone
B
b-carboline
C
Flumazenil
D
Zolpidem
High-Yield Explanation
Ans. is 'b' i.e., b-carboline Drugs acting at BZD site of GABAA receptors o Agonist at BZD site of GABAA receptor -4 Benzodiazepine, Zolpidem, Zopiclone, Zoleplon. o Inverse agonist at BZD site of GABAA receptor --> b-carboline o Competitive antagonist at BZD site of GABAA receptor ---> Flumazenil

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