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Pharmacology General Pharmacology 579309f2

Receptor agonists possess:

A
Affinity but no intrinsic activity
B
Intrinsic activity but no affinity
C
Affinity and intrinsic activity with a + sign
D
Affinity and intrinsic activity with a - sign
High-Yield Explanation
Ans. C. Affinity and intrinsic activity with a + signa. Agonist: Drug having affinity and intrinsic activity (IA)/efficacyb. Antagonist: Drug having affinity but no intrinsic activityc. Inverse agonist: Having affinity and intrinsic activity which is opposite to that of agonist e.g. beta carbolines at BDZ receptord. Partial agonist: Drug having affinity and intrinsic activity (IA)/efficacy less than agonist

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