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Pharmacology Histamine, 5-HT and PGs 538a311d

Ketoconazole should not be given to a patient being treated with astemizole because:

A
Ketoconazole induces the metabolism of astemizole
B
Dangerous ventricular arrhythmias can occur
C
Astemizole inhibits the metabolism of ketoconazole
D
Astemizole antagonizes the antifungal action of ketoconazole
High-Yield Explanation
Ketoconazole, erythromycin and clarithromycin are potent inhibitors of microsomal enzymes. Astemizole, terfenadine and cisapride are the drugs that can block cardiac K+ channels at high concentration. If administered along with microsomal enzyme inhibitors, these drugs can result in torsades de pointes, a serious polymorphic ventricular tachycardia.

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